• Title of article

    Synthesis and biological evaluation of (±)-cryptotanshinone and its simplified analogues as potent CDC25 inhibitors

  • Author/Authors

    Wei Gang Huang، نويسنده , , Ying Yan Jiang، نويسنده , , Qian Li، نويسنده , , Jia Li، نويسنده , , Jing Ya Li، نويسنده , , Wei Lu، نويسنده , , Jun Chao Cai، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2005
  • Pages
    8
  • From page
    1863
  • To page
    1870
  • Abstract
    (±)-Cryptotanshinone and its simplified analogues were synthesized via SmI2 promoted radical cyclization to construct the furan ring. Analogues and were identified as effective inhibitors of dual specificity protein phosphatase CDC25B which is a key enzyme for cell cycle progression, and they also inhibited growth in A-549 human lung cancer cell line.
  • Keywords
    Antitumor , CDC25 Inhibitor , Cryptotanshinone , Analogues
  • Journal title
    Tetrahedron
  • Serial Year
    2005
  • Journal title
    Tetrahedron
  • Record number

    1088417