• Title of article

    Free radical synthesis of benzofused tricyclic β-lactams by intramolecular cyclization of 2-azetidinone-tethered haloarenes

  • Author/Authors

    Benito Alcaide، نويسنده , , Pedro Almendros، نويسنده , , Alberto Rodr?guez-Vicente، نويسنده , , M. Pilar Ruiz، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2005
  • Pages
    12
  • From page
    2767
  • To page
    2778
  • Abstract
    o-Halogenophenyl- and o-halogenobenzyl-4-alkenyl-β-lactams can be prepared both in the racemic form and in optically pure form using the ketene–imine cyclization. These 2-azetidinone-tethered haloarenes were used for the regio- and stereoselective preparation of benzofused tricyclic β-lactams including benzocarbapenems and benzocarbacephems via intramolecular aryl radical cyclisation.
  • Keywords
    Nitrogen heterocycles , Radical reactions , Cycloaddition , polycycles , Lactams
  • Journal title
    Tetrahedron
  • Serial Year
    2005
  • Journal title
    Tetrahedron
  • Record number

    1088506