Title of article
Structure based design of simplified analogues of insect kinins
Author/Authors
Laila Kamoune، نويسنده , , Wim M. De Borggraeve، نويسنده , , Bie M.P. Verbist، نويسنده , , Jozef Vanden Broeck، نويسنده , , Geoffrey M. Coast، نويسنده , , Frans Compernolle ، نويسنده , , Georges Hoornaert، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2005
Pages
8
From page
9555
To page
9562
Abstract
Based on a receptor interaction model, simplified analogues of insect kinins were prepared. The compounds were templated on a conformationally restricted amino piperidinone carboxylate scaffold. The conformation of the analogues was studied by NMR and the biological activity of the compounds was tested in a bio-assay.
Keywords
cis-peptide bond , Insect kinin analogues
Journal title
Tetrahedron
Serial Year
2005
Journal title
Tetrahedron
Record number
1089185
Link To Document