• Title of article

    l-Proline amide-catalyzed direct asymmetric aldol reaction of aldehydes with chloroacetone

  • Author/Authors

    Long He، نويسنده , , Zhuo Tang، نويسنده , , Lin-Feng Cun، نويسنده , , Aiqiao Mi، نويسنده , , Yaozhong Jiang، نويسنده , , Liu-Zhu Gong، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2006
  • Pages
    6
  • From page
    346
  • To page
    351
  • Abstract
    l-Proline amides were evaluated for catalyzing the direct aldol reaction of 4-nitrobenzaldehyde with chloroacetone. The presence of 30 mol% (S)-pyrrolidine-2-carboxylic acid (2,4,6-trimethyl-phenyl)-amide catalyzed the direct aldol reactions of a range of aldehydes with chloroacetone to give anti-α-chloro-β-hydroxyketones with high regio-, diastereo- and enantioselectivity.
  • Keywords
    Chloroacetone , Organocatalyst , direct aldol reaction , l-proline amides , Asymmetric catalysis
  • Journal title
    Tetrahedron
  • Serial Year
    2006
  • Journal title
    Tetrahedron
  • Record number

    1089498