• Title of article

    Synthesis of pyrazino[1,2-a]benzimidazol-1(2H)ones via a microwave assisted Buchwald–Hartwig type reaction

  • Author/Authors

    Jo Alen، نويسنده , , Koen Robeyns، نويسنده , , Wim M. De Borggraeve، نويسنده , , Luc Van Meervelt، نويسنده , , Frans Compernolle ، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2008
  • Pages
    6
  • From page
    8128
  • To page
    8133
  • Abstract
    A convenient synthesis of substituted pyrazino[1,2-a]benzimidazol-1(2H)ones starting from 3,5-dichloropyrazinones has been accomplished. Various 3-anilino-pyrazinones were easily converted to the desired tricyclic structures by applying a microwave assisted Buchwald–Hartwig type cyclization.
  • Keywords
    Buchwald–Hartwig reaction , pyrazinone , Microwave chemistry
  • Journal title
    Tetrahedron
  • Serial Year
    2008
  • Journal title
    Tetrahedron
  • Record number

    1094478