• Title of article

    Copper-catalyzed tandem synthesis of [1,2,3]triazolo[5,1-a]isoquinolines and their transformation to 1,3-disubstituted isoquinolines

  • Author/Authors

    Yuanyuan Hu، نويسنده , , Jie Hu، نويسنده , , Xiang-Chuan Wang، نويسنده , , Lina Guo، نويسنده , , Xing-Zhong Shu، نويسنده , , Yan-Ning Niu، نويسنده , , Yong-Min Liang، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2010
  • Pages
    7
  • From page
    80
  • To page
    86
  • Abstract
    2-Azido-3-(2-iodophenyl)acrylates react with terminal alkynes in the presence of a copper(II) catalyst without ligands to give a wide range of [1,2,3]triazolo[5,1-a]isoquinolines in good yields. These compounds favor expulsion of N2 in refluxed acetic acid to form 1,3-disubstituted isoquinolines. The procedure is simple, economical, and efficient.
  • Journal title
    Tetrahedron
  • Serial Year
    2010
  • Journal title
    Tetrahedron
  • Record number

    1100398