• Title of article

    Tandem allylic amination/ring-opening/oxa-Michael addition reactions of chromone-derived Morita–Baylis–Hillman acetates with amines

  • Author/Authors

    Chen Wu، نويسنده , , Hao Zeng، نويسنده , , Li Liu، نويسنده , , Dong Wang، نويسنده , , Yongjun Chen، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2011
  • Pages
    7
  • From page
    1231
  • To page
    1237
  • Abstract
    The reaction of chromone-derived Morita–Baylis–Hillman acetates with amines was developed via tandem allylic amination/chromone ring-opening/oxa-Michael addition to provide 2-substituted-3-aminomethy-lene-chromans in convenient and efficient way, and subsequent applied in the synthesis of benzopyranylpyrimidine compounds. Various amines exhibited different reactivities depending on their molecular structural characteristics.
  • Keywords
    Tandom reaction , MBH acetates , Amines
  • Journal title
    Tetrahedron
  • Serial Year
    2011
  • Journal title
    Tetrahedron
  • Record number

    1102943