• Title of article

    Reaction of Tröger’s base analogues with Vilsmeier reagents

  • Author/Authors

    Qasim M. Malik، نويسنده , , Andrew B. Mahon، نويسنده , , Donald C. Craig، نويسنده , , Andrew C. Try، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2011
  • Pages
    6
  • From page
    8509
  • To page
    8514
  • Abstract
    As part of a program aimed at introducing functionality onto the Tröger’s base framework post-synthesis, we investigated the formylation reaction of Tröger’s base analogues with Vilsmeier reagents. We found that rather than the anticipated reaction at the aryl rings, these compounds react with Vilsmeier reagents to afford compounds with a modified strap, whereby the apical methylene group is replaced by a methylene strap bearing an N,N-disubstituted amine.
  • Keywords
    X-ray , Vilsmeier , Tr?ger’s base , Chirality , Bridge-modification
  • Journal title
    Tetrahedron
  • Serial Year
    2011
  • Journal title
    Tetrahedron
  • Record number

    1103812