• Title of article

    An approach to alicyclic ring-fused xanthines

  • Author/Authors

    Kostiantyn Liubchak، نويسنده , , Andrey Tolmachev، نويسنده , , Oleksandr O. Grygorenko، نويسنده , , Kostiantyn Nazarenko، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2012
  • Pages
    8
  • From page
    8564
  • To page
    8571
  • Abstract
    A convenient three-step approach to the synthesis of five to eight-membered alicyclic ring-fused xanthines was developed. The method included reaction of lactim or thiolactim ethers with 6-aminouracils, followed by bromination and copper-catalyzed arylation. The procedure allowed preparation of the title compounds in 21–36% overall yields.
  • Keywords
    Imidazoles , Amidines , Copper-catalyzed arylation , Xantines , Nitrogen Heterocycles
  • Journal title
    Tetrahedron
  • Serial Year
    2012
  • Journal title
    Tetrahedron
  • Record number

    1105018