Title of article
Lewis acid-mediated azidolysis of 2,3-three membered heterocyclic amines
Author/Authors
Giuliana Righi، نويسنده , , Giorgio Scotti، نويسنده , , Francesco Caruso، نويسنده , , Miriam Rossi، نويسنده , , Francesco Mecozzi، نويسنده , , Roberto Antonioletti، نويسنده , , Romina Pelagalli، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2013
Pages
9
From page
9557
To page
9565
Abstract
The Lewis acid-catalyzed regioselective azidolysis of 2,3-three membered heterocyclic amines has been investigated. The results obtained demonstrated that using TMSN3 as a source of azide, the appropriate choice of Lewis acid allowed to obtain different regio- and stereocontrolled precursors of aminoalcoholic and triaminic sequences. Considering the occurrence of these moieties in the structure of many biologically active compounds, the present methodologies could represent a powerful tool in organic synthesis for the preparation of interesting molecules.
Journal title
Tetrahedron
Serial Year
2013
Journal title
Tetrahedron
Record number
1106414
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