• Title of article

    Acid-Mediated Highly Regioselective Oxidation of Substituted Furans: A Simple and Direct Entry to Substituted Butenolides

  • Author/Authors

    Cenal، Juan P. نويسنده , , Carreras، Carlos R. نويسنده , , Tonn، Carlos E. نويسنده , , Padron، Juan I. نويسنده , , Ramirez، Miguel A. نويسنده , , Diaz، David D. نويسنده , , Garcia-Tellado، Fernando نويسنده , , Martin، Victor S. نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2005
  • Pages
    -1574
  • From page
    1575
  • To page
    0
  • Abstract
    The scope and limitations of an expeditious synthesis of substituted butenolides from 3-substituted or 3,4-disubstituted furans is described. The entire process embodies a controlled oxidation of the furan core to a 2,5dialkoxy-dihydrofuran intermediate and a regioselective acid-catalyzed hydrolysis to the butenolide derivative. 3-Substituted furans yield exclusively 2-substituted butenolides. Calculations studies provide substantiation of a proposed mechanism.
  • Keywords
    substituted butenolides , Furans , Oxidation
  • Journal title
    Synlett
  • Serial Year
    2005
  • Journal title
    Synlett
  • Record number

    110697