• Title of article

    Synthesis of 4,5-difluoroimidazole

  • Author/Authors

    Dolensky، نويسنده , , Bohumil and Takeuchi، نويسنده , , Yoshio and Cohen، نويسنده , , Louis A and Kirk، نويسنده , , Kenneth L، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2001
  • Pages
    2
  • From page
    147
  • To page
    148
  • Abstract
    5-Fluoroimidazole-4-carboxylic acid ethyl ester was converted to the corresponding hydrazide. Oxidation of the hydrazide to the carbonyl azide and Curtius rearrangement in t-butyl alcohol produced 4-t-butyloxycarbonylamino-5-fluoroimidazole. Dissolution of the t-butyl carbamate in 50% HBF4, in situ diazotation of the resulting amine, and irradiation produced the target compound.
  • Keywords
    Photochemical Schiemann reaction , Fluoroimidazoles
  • Journal title
    Journal of Fluorine Chemistry
  • Serial Year
    2001
  • Journal title
    Journal of Fluorine Chemistry
  • Record number

    1603049