• Title of article

    Asymmetric synthesis of the key intermediate of an SP antagonist RPR107880 using a base-catalyzed Diels–Alder reaction

  • Author/Authors

    Okamura، نويسنده , , Hiroaki and Shimizu، نويسنده , , Hideki and Nakamura، نويسنده , , Yasuko and Iwagawa، نويسنده , , Tetsuo and Nakatani، نويسنده , , Munehiro، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2000
  • Pages
    4
  • From page
    4147
  • To page
    4150
  • Abstract
    An asymmetric synthesis of the key intermediate of RPR 107880, a substance P antagonist, using a base-catalyzed Diels–Alder reaction of 3-hydroxy-2-pyrone and N-benzylmaleimide is described.
  • Keywords
    base-catalyzed Diels–Alder reaction , asymmetric synthesis , substance P , RPR 107880
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2000
  • Journal title
    Tetrahedron Letters
  • Record number

    1637781