• Title of article

    Solid phase synthesis of peptide vinyl sulfone and peptide epoxyketone proteasome inhibitors

  • Author/Authors

    Overkleeft، نويسنده , , Herman S and Bos، نويسنده , , Pepijn R and Hekking، نويسنده , , Brian Francis and Gordon Harris، نويسنده , , Eva J and Ploegh، نويسنده , , Hidde L and Kessler، نويسنده , , Benedikt M، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2000
  • Pages
    5
  • From page
    6005
  • To page
    6009
  • Abstract
    The solid phase synthesis of the known proteasome inhibitor ZL3VS, using Kennerʹs safety catch protocol, is described. This methodology has been extended to the synthesis of various novel peptide vinyl sulfone and peptide epoxyketone derivatives.
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2000
  • Journal title
    Tetrahedron Letters
  • Record number

    1638343