• Title of article

    Total synthesis and biological evaluation of apicularen A and synthetic analogs

  • Author/Authors

    Bhattacharjee، نويسنده , , Ashoke and Seguil، نويسنده , , Olga R and De Brabander، نويسنده , , Jef K، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2001
  • Pages
    4
  • From page
    1217
  • To page
    1220
  • Abstract
    The first total synthesis of the potent cytostatic agent apicularen A is described along with the synthesis of the corresponding C11-epimers and side chain modified congeners. Growth inhibition experiments with the human melanoma cancer cell line SK-MEL-5 revealed an important role for the unusual N-acyl enamide side chain.
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2001
  • Journal title
    Tetrahedron Letters
  • Record number

    1641869