Title of article
A novel method for the mild and selective amidation of diesters and the amidation of monoesters
Author/Authors
Guo، نويسنده , , Zhenrong and Dowdy، نويسنده , , Eric D and Li، نويسنده , , Wen-Sen and Polniaszek، نويسنده , , Richard and Delaney، نويسنده , , Edward، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2001
Pages
3
From page
1843
To page
1845
Abstract
The selective monoamidation of diesters and amidation of esters mediated by Lewis acids are described. The selective amidations of dimethyl pyridine-2,5-dicarboxylate (1) and dimethyl 2,3-indole-dicarboxylate (4) with primary and secondary amines mediated by MgCl2 or MgBr2 under mild conditions gave the corresponding ester-amides in high yield.
Keywords
selective amidation of diesters , amidation of esters , Lewis acids
Journal title
Tetrahedron Letters
Serial Year
2001
Journal title
Tetrahedron Letters
Record number
1643535
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