• Title of article

    Sonogashira cross-coupling reaction of 3-iodoindazoles with various terminal alkynes: a mild and flexible strategy to design 2-aza tryptamines

  • Author/Authors

    M. Zaharia-Arnautu، نويسنده , , Anca and Collot، نويسنده , , Valérie and Ros، نويسنده , , Javier Calvo and Alayrac، نويسنده , , Carole and Witulski، نويسنده , , Bernhard and Rault، نويسنده , , Sylvain، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2002
  • Pages
    3
  • From page
    2695
  • To page
    2697
  • Abstract
    This paper describes a Sonogashira-type cross-coupling reaction of 3-iodoindazoles with various terminal alkynes as a general route to 3-alkynylindazoles. The coupling reaction is illustrated by the preparation of new indazolylpropiolic or propargylic derivatives. Scope and limitation of the method are outlined.
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2002
  • Journal title
    Tetrahedron Letters
  • Record number

    1650988