Title of article
A simple, two-step synthesis of 3-iodoindoles
Author/Authors
Amjad، نويسنده , , Muhammad and Knight، نويسنده , , David W.، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2004
Pages
3
From page
539
To page
541
Abstract
2-Halo-anilines, protected as the corresponding sulfonamides or carbamates, can be converted very efficiently into 3-iodoindoles by sequential Sonogashira coupling with a 1-alkyne and 5-endo-dig iodocyclisation. Azaindoles can also be obtained using this methodology.
Keywords
5-endo-dig , indole , Synthesis , iodocyclisation , Sonogashira
Journal title
Tetrahedron Letters
Serial Year
2004
Journal title
Tetrahedron Letters
Record number
1656521
Link To Document