• Title of article

    Palladium-catalysed amination of 2-acyl-1-alkyl-5-bromopyrroles

  • Author/Authors

    Castellote، نويسنده , , Isabel and Vaquero، نويسنده , , Juan J. and Alvarez-Builla، نويسنده , , Julio، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2004
  • Pages
    4
  • From page
    769
  • To page
    772
  • Abstract
    The first intermolecular C–N bond-forming reactions between substituted 2-bromopyrroles and primary and cyclic secondary amines were performed using Pd2(dba)3 as catalyst with BINAP as the ligand. The aminations proceeded in the presence of NaOtBu at 80–100 °C in 31–93% yields.
  • Keywords
    PALLADIUM , Catalysed , Functionalised , 2-Halopyrroles , amination
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2004
  • Journal title
    Tetrahedron Letters
  • Record number

    1656672