• Title of article

    Preparation of N-hydroxysuccinimido esters via palladium-catalyzed carbonylation of aryl triflates and halides

  • Author/Authors

    Lou، نويسنده , , Rongliang and VanAlstine، نويسنده , , Melissa and Sun، نويسنده , , Xufeng and Wentland، نويسنده , , Mark P.، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2003
  • Pages
    4
  • From page
    2477
  • To page
    2480
  • Abstract
    N-Hydroxysuccinimido esters of aromatic carboxylic acids (a.k.a. active esters) can be made using a potentially general, one-step procedure via Pd-catalyzed carbonylation of an aryl triflate or aryl iodide with CO and N-hydroxysuccinimide. Excellent yields (up to 94%) were observed when the reaction was done in DMSO at 70°C and 1 atmosphere of CO pressure.
  • Keywords
    N-hydroxysuccinimide , Pd-catalyzed carbonylation , Active ester
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2003
  • Journal title
    Tetrahedron Letters
  • Record number

    1661277