• Title of article

    Synthesis of (±)-solanapyrones A and B

  • Author/Authors

    Lygo، نويسنده , , Barry and Bhatia، نويسنده , , Mohamed and Cooke، نويسنده , , Jason W.B. and Hirst، نويسنده , , David J.، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2003
  • Pages
    4
  • From page
    2529
  • To page
    2532
  • Abstract
    In this paper we report the development of a stereoselective IMDA approach to the phytotoxic polyketides (±)-solanapyrones A and B. The stereoselectivity of the key IMDA cycloaddition was optimized by investigating a range of 2,8,10-dodecatrienoic acid derivatives. This established that use of the Weinreb amide led to the desired exo-selectivity and also facilitated construction of the pyrone moiety. A novel approach to the installation of the C-3 formyl group in solanapyrone A is also described.
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2003
  • Journal title
    Tetrahedron Letters
  • Record number

    1661314