Title of article
New potent insecticidal agent: 4′-fucosyl avermectin derivative
Author/Authors
Wei، نويسنده , , Guohua and Du، نويسنده , , Yuguo and Linhardt، نويسنده , , Robert J.، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2004
Pages
4
From page
6895
To page
6898
Abstract
A 4′-fucosyl avermectin derivative was designed and synthesized. This new avermectin derivative showed excellent in vivo bioactivity against cabbage larvae when compared to commercially available avermectin B1a. In this synthesis, thioglycosyl donors, but not trichloroacetimidates, were found compatible with sugar-macrolide synthesis under rt promotion with NIS or I2 in N-methylpyrrolidone.
Keywords
Synthesis , glycosylation , Insecticide , Avermectin , Fucosyl avermectin
Journal title
Tetrahedron Letters
Serial Year
2004
Journal title
Tetrahedron Letters
Record number
1843202
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