• Title of article

    Expedient synthesis of 1-vinylpyrrole-2-carbaldehydes

  • Author/Authors

    Mikhaleva، نويسنده , , Al’bina I. and Zaitsev، نويسنده , , Alexey B. and Ivanov، نويسنده , , Andrey V. and Schmidt، نويسنده , , Elena Yu. and Vasilʹtsov، نويسنده , , Alexander M. and Trofimov، نويسنده , , Boris A.، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2006
  • Pages
    4
  • From page
    3693
  • To page
    3696
  • Abstract
    1-Vinylpyrrole-2-carbaldehydes and 1-vinyl-4,5-dihydrobenzo[g]indole-2-carbaldehyde were synthesized in 56–91% yields from their 1-vinyl derivatives by a modified Vilsmeier–Haack reaction. A low temperature (−78 °C) is required to avoid removal of the N-vinyl group, whereas at elevated temperature (reflux in 1,2-dichloroethane) the latter process leads to direct conversion of 1-vinylpyrroles to pyrrole-2-carbaldehydes.
  • Keywords
    1-Vinylpyrrole , 1-Vinylpyrrole-2-carbaldehydes , Formylation , Vilsmeier–Haack reaction
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2006
  • Journal title
    Tetrahedron Letters
  • Record number

    1850432