Title of article
Asymmetric induction in the reactions of 3-aryl-1,2,4-triazin-5(4H)-ones with C-nucleophiles
Author/Authors
Egorov، نويسنده , , Ilya N. and Zyryanov، نويسنده , , Grigory V. and Ulomsky، نويسنده , , Eugeny N. and Rusinov، نويسنده , , Vladimir L. and Chupakhin، نويسنده , , Oleg N.، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2006
Pages
3
From page
7485
To page
7487
Abstract
3-Aryl-1,2,4-triazin-5(4H)-ones, in the presence of N-protected amino acids, react with C-nucleophiles to form 1-acyl-6-Nu-3-aryl-1,6-dihydro-1,2,4-triazin-5(4H)-ones in high diastereomeric excess. This is the first case of the use of amino acids as chiral auxiliaries in nucleophilic additions to triazinones.
Journal title
Tetrahedron Letters
Serial Year
2006
Journal title
Tetrahedron Letters
Record number
1852837
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