Title of article
A novel palladium catalyst for the amination of electron-rich indole derivatives
Author/Authors
Schwarz، نويسنده , , Nicolle and Tillack، نويسنده , , Annegret and Alex، نويسنده , , Karolin and Sayyed، نويسنده , , Iliyas Ali and Jackstell، نويسنده , , Ralf and Beller، نويسنده , , Matthias، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2007
Pages
4
From page
2897
To page
2900
Abstract
The palladium-catalyzed amination of a 3-silyloxy-substituted bromo-indole with primary and secondary amines is described for the first time. In the presence of the novel catalyst system of Pd(OAc)2/N-phenyl-2-(di-1-adamantylphosphino)pyrrole potentially bioactive amino-functionalized indole derivatives are obtained in a general manner in high yield.
Keywords
amination , C–N coupling , PALLADIUM , indoles
Journal title
Tetrahedron Letters
Serial Year
2007
Journal title
Tetrahedron Letters
Record number
1854776
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