• Title of article

    An efficient synthesis of 4-bromo-N-substituted oxindoles by an intramolecular copper-catalyzed amidation reaction

  • Author/Authors

    van den Hoogenband، نويسنده , , Adri and Lange، نويسنده , , Jos H.M. and den Hartog، نويسنده , , Jack A.J. and Henzen، نويسنده , , Remco and Terpstra، نويسنده , , Jan Willem، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2007
  • Pages
    5
  • From page
    4461
  • To page
    4465
  • Abstract
    A highly efficient synthetic approach to novel 4-bromo-N-substituted oxindoles is described. The method involves a mild intramolecular copper-catalyzed amidation reaction of N-substituted 2,6-dibromophenylacetamides. In contrast to our recently published palladium-catalyzed amidation reaction, no concomitant dimerization on the 3-position of the formed oxindole occurs.
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2007
  • Journal title
    Tetrahedron Letters
  • Record number

    1855306