Title of article
One-pot synthesis of β-imidazolylpropionamides
Author/Authors
Sergey V. Ryabukhin، نويسنده , , Sergey V. and Granat، نويسنده , , Dmitry S. and Khodakovskiy، نويسنده , , Pavel V. and Shivanyuk، نويسنده , , Alexander N. and Tolmachev، نويسنده , , Andrey A.، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2008
Pages
6
From page
3997
To page
4002
Abstract
New efficient one-pot methodology for the preparative synthesis of β-imidazolylpropionamides was elaborated. It is based on the addition of imidazole to the activated double bond of the intermediate acrylimidazolide in the reaction between diverse acrylic acids and different amines promoted by CDI. A set of structurally and functionally diverse β-imidazolylpropionamides was obtained in high preparative yields.
Keywords
Acrylic acids , ?-Imidazolylpropionamides , Carbonyldiimidazole (CDI) , acylation
Journal title
Tetrahedron Letters
Serial Year
2008
Journal title
Tetrahedron Letters
Record number
1859561
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