Title of article
Aminomethylation of lithiated nicotinamide: access to new pyridolactams
Author/Authors
Prieur، نويسنده , , Emilie and Azzouz، نويسنده , , Rabah and Deguest، نويسنده , , Geoffrey and Fruit، نويسنده , , Corinne and Bischoff، نويسنده , , Laurent and Marsais، نويسنده , , Francis، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2008
Pages
4
From page
437
To page
440
Abstract
New 2,3-dihydropyrrolopyridinones were conveniently prepared by trapping lithiated pyridine carboxamides with highly reactive formimines. In this Letter, we report that a wide range of N-functionalised compounds can be synthesised in one step by this process, allowing the presence of ethers, acetals or ester moieties.
Keywords
pyridine , Lactam , Aminomethylation , Formimine , Metalation
Journal title
Tetrahedron Letters
Serial Year
2008
Journal title
Tetrahedron Letters
Record number
1860032
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