• Title of article

    Asymmetric cycloetherification based on a chiral auxiliary for 4-acyloxy-1-butene substrates during oxidation with iodosylbenzene via a 1,3-dioxan-2-yl cation

  • Author/Authors

    Fujita، نويسنده , , Morifumi and Ookubo، نويسنده , , Yuuya and Sugimura، نويسنده , , Takashi، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2009
  • Pages
    3
  • From page
    1298
  • To page
    1300
  • Abstract
    Reaction of but-3-enyl camphanate and its derivatives with iodosylbenzene yielded tetrahydrofuran-3-yl camphanate with high diastereomeric ratio via a 1,3-dioxan-2-yl cation intermediate. The reaction using (1S)-camphanate as a chiral auxiliary preferentially gave (S)-3-acyloxytetrahydrofuran and (2S,3S)-3-acyloxy-2-silyltetrahydrofuran.
  • Keywords
    Neighboring group participation , Iodosylbenzene , Tetrahydrofuran , hypervalent iodine , chiral auxiliary
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2009
  • Journal title
    Tetrahedron Letters
  • Record number

    1862906