• Title of article

    Highly cis- and trans-selective alkyl radical addition to α-methylene-γ-phenyl-γ-butyrolactams

  • Author/Authors

    Yajima، نويسنده , , Tomoko and Hamano، نويسنده , , Masako and Nagano، نويسنده , , Hajime، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2009
  • Pages
    2
  • From page
    1301
  • To page
    1302
  • Abstract
    The 1,3-asymmetric induction in alkyl radical additions to α-methylene-γ-phenyl-γ-butyrolactams was investigated. The reactions of N-unsubstituted lactam using (Me3Si)3SiH under UV irradiation give cis-α,γ-disubstituted lactams, whereas reactions of N-pivaloyllactams using Et3B and Bu3SnH in the presence of Yb(OTf)3 give trans-α,γ-disubstituted lactams, both with high diastereoselectivities.
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2009
  • Journal title
    Tetrahedron Letters
  • Record number

    1862907