Title of article
NIS-promoted guanylation of amines
Author/Authors
Ohara، نويسنده , , Keiichiro and Vasseur، نويسنده , , Jean-Jacques and Smietana، نويسنده , , Michael، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2009
Pages
3
From page
1463
To page
1465
Abstract
An efficient NIS-promoted guanylation reaction is described. This procedure allows the guanylation of primary and secondary amines through the reaction with di-Boc-thiourea and di-Boc-S-methylisothiourea, respectively. We demonstrated that the use of NIS compares favorably with existing methods and is an attractive alternative to heavy metal or Mukayama’s reagent activation.
Keywords
Guanidine , Thiourea derivatives , NIS
Journal title
Tetrahedron Letters
Serial Year
2009
Journal title
Tetrahedron Letters
Record number
1862987
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