• Title of article

    Selective phenol alkylation for an improved synthesis of 2-arylbenzimidazole H4 receptor ligands

  • Author/Authors

    Savall، نويسنده , , Brad M. and Fontimayor، نويسنده , , Jill R. and Edwards، نويسنده , , James P.، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2009
  • Pages
    3
  • From page
    2490
  • To page
    2492
  • Abstract
    Alkylation of a phenol OH in the presence of a free benzimidazole NH was investigated and found to be highly dependent on the substitution of the benzimidazole and phenol rings. The modification of our original synthesis of 2-arylbenzimidazole H4 receptor ligands has resulted in improved yields and ease of isolation of final products.
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2009
  • Journal title
    Tetrahedron Letters
  • Record number

    1863716