• Title of article

    Intramolecular amidocyclopropanation reactions using diethoxymethyl-functionalised lactams as organozinc carbenoid precursors

  • Author/Authors

    Jerome، نويسنده , , Laure and Sheppard، نويسنده , , Tom D. and Aliev، نويسنده , , Abil E. and Motherwell، نويسنده , , William B.، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2009
  • Pages
    4
  • From page
    3709
  • To page
    3712
  • Abstract
    Intramolecular amidocyclopropanation reactions of diethoxymethyl-lactams containing a pendant alkene were examined using zinc/TMSCl. With a range of 4–6-membered lactams, bicyclic amidocyclopropanes were obtained with very high diastereoselectivity with a preference for the formation of the more hindered endo-cyclopropane.
  • Keywords
    carbenoids , lactams , Cyclopropanes , Zinc , alkenes
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2009
  • Journal title
    Tetrahedron Letters
  • Record number

    1864631