Title of article
Palladium-catalyzed benzylation of N-Boc indole boronic acids
Author/Authors
Kearney، نويسنده , , Aaron M. and Landry-Bayle، نويسنده , , Adrienne and Gomez، نويسنده , , Laurent، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2010
Pages
3
From page
2281
To page
2283
Abstract
The direct benzylation of indole 2-boronic acid can be efficiently achieved using trans-PdBr(N-Succ)(PPh3)2, alleviating the need for strong bases or toxic organotin reagents. Under these reaction conditions substituted indole-2-boronic acids and substituted benzyl bromides are cross-coupled to afford aryl(indolo)methanes in good yield.
Journal title
Tetrahedron Letters
Serial Year
2010
Journal title
Tetrahedron Letters
Record number
1872043
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