• Title of article

    Synthesis of a tricyclic core of rameswaralide

  • Author/Authors

    Trost، نويسنده , , Barry M. and Nguyen، نويسنده , , Hien M. and Koradin، نويسنده , , Christopher، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2010
  • Pages
    4
  • From page
    6232
  • To page
    6235
  • Abstract
    A tricyclic core containing a 5,7-fused bicyclic unit of rameswaralide was prepared starting from a 1,6-enyne. The synthetic sequence involved (i) ruthenium-catalyzed [5+2]-cycloaddition of 1,6-enyne, (ii) an acyl radical based approach to construct the lactone, and (iii) a regioselective installation of the conjugated double bond by a concomitant sulfenylation–dehydrosulfenylation sequence.
  • Keywords
    The fused bicyclic system , reductive radical cyclization , total synthesis , cycloaddition , Ruthenium
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2010
  • Journal title
    Tetrahedron Letters
  • Record number

    1875647