• Title of article

    Synthesis of fused dihydropyrido[e]purines via ring closing metathesis

  • Author/Authors

    Litinas، نويسنده , , Konstantinos E. and Thalassitis، نويسنده , , Andreas، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2010
  • Pages
    3
  • From page
    6451
  • To page
    6453
  • Abstract
    Ring closing metathesis (RCM) of 8,9-diallylpurines or 9-butenyl-8-vinylpurines with the Grubbs 2nd generation catalyst resulted in fused 6,9- or 8,9-dihydropyrido[e]purines, respectively. The 8,9-dialkenylpurines were prepared from 8-bromopurines after 9-alkenylation and subsequent Stille coupling at C-8 with alkenylstannanes in the presence of Pd(PPh3)4 or Pd(PPh3)2Cl2.
  • Keywords
    Ring closing metathesis , Stille coupling , Pd(PPh3)4
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2010
  • Journal title
    Tetrahedron Letters
  • Record number

    1875822