• Title of article

    Sequential alkylation/gold-catalyzed annulation reactions of anilines with propargylic bromide derivatives

  • Author/Authors

    Alfonsi، نويسنده , , Maria and Arcadi، نويسنده , , Antonio and Chiarini، نويسنده , , Marco and Marinelli، نويسنده , , Fabio، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2011
  • Pages
    4
  • From page
    5145
  • To page
    5148
  • Abstract
    Preliminary results of sequential alkylation/gold-catalyzed annulation reactions of anilines with propargylic bromide derivatives to provide quinoline scaffolds are described. The efficiency of NaAuCl4·2H2O in the sequential procedure was investigated and compared with different transition metal salts and Au(I) complexes. Selectivity of the reaction of aniline derivatives with propargylic bromides has also been investigated.
  • Keywords
    Sequential reactions , gold catalysis , N-Propargylation , Quinolines , Intramolecular hydroarylation
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2011
  • Journal title
    Tetrahedron Letters
  • Record number

    1879312