• Title of article

    Stereoselective synthesis of analogs of the macrolactone of isomigrastatin

  • Author/Authors

    Dias، نويسنده , , Luiz C. and Monteiro، نويسنده , , Gustavo C. and Amarante، نويسنده , , Giovanni W. and Conegero، نويسنده , , Leila S. and Finelli، نويسنده , , Fernanda G.، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2012
  • Pages
    3
  • From page
    707
  • To page
    709
  • Abstract
    An approach for the highly stereoselective synthesis of analogs of the macrolactone of isomigrastatin is described. Our optimized strategy is based on a very efficient lactone opening, a Wittig olefination reaction and a ring closing metathesis. The syntheses were accomplished in 10–11 steps and good overall yields.
  • Keywords
    Dihydroxilation reaction , Ring closing metathesis , macrolactone , Tumor metastasis , Migrastatin
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2012
  • Journal title
    Tetrahedron Letters
  • Record number

    1880076