• Title of article

    Olefin cross-metathesis/Suzuki–Miyaura reactions on vinylphenylboronic acid pinacol esters

  • Author/Authors

    Baltus، نويسنده , , Christine B. and Chuckowree، نويسنده , , Irina S. and Press، نويسنده , , Neil J. and Day، نويسنده , , Iain J. and Coles، نويسنده , , Simon J. and Tizzard، نويسنده , , Graham J. and Spencer، نويسنده , , John، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2013
  • Pages
    7
  • From page
    1211
  • To page
    1217
  • Abstract
    A series of alkenyl phenylboronic acid pinacol esters has been synthesized via an olefin cross-metathesis reaction of vinylphenylboronic acid pinacol ester derivatives. After catalytic hydrogenation, the resulting boronates were coupled via a microwave-mediated Suzuki–Miyaura reaction to afford a library of biarylethyl aryl and biarylethyl cycloalkyl derivatives. A complementary reaction sequence involved an initial Suzuki–Miyaura coupling.
  • Keywords
    Arylboronic esters , cross-metathesis , C–C bond formation , Microwaves , Suzuki–Miyaura coupling
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2013
  • Journal title
    Tetrahedron Letters
  • Record number

    1883868