• Title of article

    Synthesis of pyrazolo[1,5-a]pyridines by thermal intramolecular cyclization

  • Author/Authors

    Hoashi، نويسنده , , Yasutaka and Takai، نويسنده , , Takafumi and Kotani، نويسنده , , Etsuo and Koike، نويسنده , , Tatsuki، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2013
  • Pages
    4
  • From page
    2199
  • To page
    2202
  • Abstract
    Thermal intramolecular cyclization of N-amino-2-alkynylpyridines was developed for facile and versatile synthesis of pyrazolo[1,5-a]pyridines. Simply heating N-amino-2-alkynylpyridines in acetic acid provided pyrazolo[1,5-a]pyridines in excellent yield.
  • Keywords
    Thermal intramolecular cyclization , Melatonin receptor agonist , 5-a]pyridine , N-Amino-2-alkynylpyridine
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2013
  • Journal title
    Tetrahedron Letters
  • Record number

    1884280