• Title of article

    Metal-free 5-exo-dig cyclization of propargyl urea using TBAF

  • Author/Authors

    Huguenot، نويسنده , , Florent and Delalande، نويسنده , , Clémence and Vidal، نويسنده , , Michel، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2014
  • Pages
    4
  • From page
    4632
  • To page
    4635
  • Abstract
    We present the first results of the intramolecular cyclization of propargyl ureas catalyzed by TBAF. Depending on the substituents close to the triple bond, imidazolone or methylene-imidazolidinone was obtained. The dual activation of the triple bond by interaction with TBAF via the cation–π is thought to be responsible.
  • Keywords
    Propargyl urea , Intermolecular cyclization , TBAF , cation–? interaction , Imidazolinone
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2014
  • Journal title
    Tetrahedron Letters
  • Record number

    1890388