Title of article
Protein kinase C-α inhibitors; structure-activity relationships in bis-indole series
Author/Authors
Guojian Xie، نويسنده , , Jürg Zimmermann، نويسنده , , Thomas Meyer، نويسنده , , J. William Lown، نويسنده ,
Issue Information
روزنامه با شماره پیاپی سال 1995
Pages
4
From page
497
To page
500
Abstract
To assess the role of the amine and ester containing oligopeptide side-chains in bis-indole protein kinase C inhibitors, six novel hybrids in this series were synthesized. These new compounds displayed effective inhibitory activity against protein kinase C-α.
Journal title
Bioorganic & Medicinal Chemistry Letters
Serial Year
1995
Journal title
Bioorganic & Medicinal Chemistry Letters
Record number
787361
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