• Title of article

    Glycomimetic selectin inhibitors: (α-D-mannopyranosyloxy)methylbiphenyls

  • Author/Authors

    Brian Dupré، نويسنده , , Huong Bui، نويسنده , , Ian L. Scott، نويسنده , , Robert V. Market، نويسنده , , Karin M. Keller، نويسنده , , Pamela J. Beck، نويسنده , , Timothy P. Kogan، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 1996
  • Pages
    4
  • From page
    569
  • To page
    572
  • Abstract
    A novel class of biphenyl-based compounds were investigated for their ability to inhibit sialyl Lewis X (sLex) dependent binding of HL-60 cells to E- and P-selectin fusion proteins. Compounds ( ) and ( ) demonstrated improved binding as compared to both the natural ligand sLex and a previously reported inhibitor TBC-265 ( , R = 3-CH2CO2H).
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    1996
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    787959