• Title of article

    Synthesis and in vitro cytotoxicity of cryptophycins and related analogs

  • Author/Authors

    Jean-Marc de Muys، نويسنده , , Rabindra Rej، نويسنده , , Dieu Nguyen، نويسنده , , Brian Go، نويسنده , , Samuel Fortin، نويسنده , , Jean-François Lavallée، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 1996
  • Pages
    6
  • From page
    1111
  • To page
    1116
  • Abstract
    Several members of the Cryptophycin family were synthesised using a straightforward convergent approach. The proposed synthetic route was used to prepare novel analogs of Cryptophycins A and B in which the benzylic epoxide moiety was replaced by alternate electrophilic functions. The effect of these modifications on cytotoxic activity was determined on several tumor cell lines.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    1996
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    788069