• Title of article

    Conformationally restricted 1,5-diarylpyrazoles are selective COX-2 inhibitors

  • Author/Authors

    Stephen R. Bertenshaw، نويسنده , , John J. Talley، نويسنده , , D.J. Rogier، نويسنده , , Matthew J. Graneto، نويسنده , , Carol M. Koboldt، نويسنده , , Yan Zhang، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 1996
  • Pages
    4
  • From page
    2827
  • To page
    2830
  • Abstract
    Benzothiopyranopyrazoles and benzopyranopyrazoles containing either a sulfone or sulfonamide moiety were synthesized and tested for COX-1 and COX-2 inhibition. This new class of COX-2 selective inhibitors possess antiinflammatory activity in vivo.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    1996
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    788448