• Title of article

    Synthesis and antitumor activity of leinamycin derivatives: Modifications of C-8 hydroxy and C-9 keto groups

  • Author/Authors

    Yutaka Kanda، نويسنده , , Tadashi Ashizawa، نويسنده , , Yutaka Saitoh، نويسنده , , Hiromitsu Saito، نويسنده , , Katsushige Gomi، نويسنده , , Masami Okabe، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 1998
  • Pages
    4
  • From page
    909
  • To page
    912
  • Abstract
    A series of leinamycin derivatives were synthesized and evaluated for antitumor activity. Modifications at C-8 and C-9 positions revealed a broad structure-activity relationship in vitro and some derivatives showed potent antiproliferative activity against HeLa S3 cells.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    1998
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    789346