• Title of article

    Synthesis of -enantiomers of 4′-thioarabinofuranosyl pyrimidine nucleosides

  • Author/Authors

    Hiroshi Satoh، نويسنده , , Yuichi Yoshimura، نويسنده , , Shinji Sakata، نويسنده , , Shinji Miura، نويسنده , , Haruhiko Machida، نويسنده , , Akira Matsuda and Fuyuhiko Inagaki، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 1998
  • Pages
    4
  • From page
    989
  • To page
    992
  • Abstract
    -Enantiomers of 4′-thioarabinofuranosyl pyrimidine nucleosides were synthesized from -xylose. Methyl 6 was converted to the corresponding xylitol 7, which was treated with MsCl and then Na2S to give 1,4-anhydro- -4-thioarabitol 8. As previously reported, Pummerer rearrangement of 8 followed by glycosylation with a silylated thymine and N4-acetylcytosine derivative and deprotection gave the corresponding α- and β- -4′-thioarabinofuranosyl pyrimidine nucleosides.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    1998
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    789362