• Title of article

    Anti-inflammatory/antiarthritic ketonic bisphosphonic acid esters

  • Author/Authors

    Stephen T. Schlachter، نويسنده , , Louise A. Galinet، نويسنده , , Sharon K. Shields، نويسنده , , Danielle G. Aspar، نويسنده , , Colin J. Dunn، نويسنده , , Nigel D. Staite، نويسنده , , Richard A. Nugent، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 1998
  • Pages
    4
  • From page
    1093
  • To page
    1096
  • Abstract
    Bisphosphonate ester 2 is an inhibitor of inflammation, but is devoid of antiarthritic effects. SAR studies on a series of related bisphosphonate esters resulted in compounds 6e, 6i, 6j, and 6m, which exhibited excellent inhibition of an arthritis model, in addition to potent anti-inflammatory effects.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    1998
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    789382