• Title of article

    SAR studies of diaryltriazoles against bacterial two-component regulatory systems and their antibacterial activities

  • Author/Authors

    Zhihua Sui، نويسنده , , Jihua Guan، نويسنده , , Dennis J. Hlasta، نويسنده , , Mark J. Macielag، نويسنده , , Barbara D. Foleno، نويسنده , , Raul M. Goldschmidt، نويسنده , , Michael J. Loeloff، نويسنده , , Glenda C. Webb، نويسنده , , John F. Barrett، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 1998
  • Pages
    6
  • From page
    1929
  • To page
    1934
  • Abstract
    A series of diaryltriazole analogs was discovered to inhibit bacterial two-component regulatory systems in our primary assays, KinA/SpoOF and NRII/NRI. They also showed inhibitory activity in whole cell mechanism-based assays, and they possessed potent activities against several strains of Gram-positive pathogenic bacteria in the standard MIC broth assay.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    1998
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    789546