• Title of article

    Synthetic oligosaccharides having various functional domains: Potent and potentially safe heparin mimetics

  • Author/Authors

    Maurice Petitou، نويسنده , , Pierre Alexandre Driguez، نويسنده , , Philippe Duchaussoy، نويسنده , , Jean-Pascal Hérault، نويسنده , , Jean-Claude Lormeau، نويسنده , , Jean-Marc Herbert، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 1999
  • Pages
    6
  • From page
    1161
  • To page
    1166
  • Abstract
    A synthetic heptadecasaccharide, comprising an antithrombin III binding domain, a thrombin binding domain, and a neutral methylated hexasaccharide sequence, was obtained through a convergent synthesis. This compound displayed in vitro anticoagulant properties similar to that of standard heparin but, in contrast with heparin, escaped neutralization by platelet factor 4, a protein released by activated platelets.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    1999
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    790111